Discovery and Optimization of a Novel Series of Highly Selective JAK1 Kinase Inhibitors.
Neil P Grimster,Erica Anderson,Marat Alimzhanov,Geraldine Bebernitz,Kirsten Bell,Claudio Chuaqui,Tracy Deegan,Andrew D Ferguson,Thomas Gero,Andreas Harsch,Dennis Huszar,Aarti Kawatkar,Jason G Kettle,Paul Lyne,Jon A Read,Caroline Rivard Costa,Linette Ruston,Patricia Schroeder,Jie Shi,Qibin Su,Scott Throner,Dorin Toader,Melissa Vasbinder,Richard Woessner,Haixia Wang,Allan Wu,Minwei Ye,Weijia Zheng,Michael Zinda JOURNAL OF MEDICINAL CHEMISTRY(2018)
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