Discovery of (2R)-N-[3-[2-[(3-Methoxy-1-methyl-pyrazol-4-yl)amino]pyrim idin-4-yl]-1H-indol-7-yl]-2-(4-methylpiperazin-1-yl)propenamide (AZD4205) as a Potent and Selective Janus Kinase 1 InhibitorQibin Su,Erica Banks,Geraldine Bebernitz,Kirsten Bell, Cassandra F. Borenstein,Huawei Chen, Claudio E. Chuaqui,Nanhua Deng,Andrew D. Ferguson,Sameer Kawatkar,Neil P. Grimster,Linette Ruston,Paul D. Lyne,Jon A. Read, Xianyou Peng,Xiaohui Pei,Stephen Fawell, Zhanlei Tang,Scott Throner,Melissa M. Vasbinder,Haoyu Wang,Jon Winter-Holt,Richard Woessner,Allan Wu,Wenzhan Yang,Michael Zinda,Jason G. KettleJOURNAL OF MEDICINAL CHEMISTRY(2020)引用 0|浏览2AI 理解论文溯源树样例生成溯源树,研究论文发展脉络Chat Paper正在生成论文摘要