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An Efficient Site-Selective, Dual Bioconjugation Approach Exploiting N-terminal Cysteines As Minimalistic Handles to Engineer Tailored Anti-Her2 Affibody Conjugates

Ana Novak, Florian Kersaudy,Sylvie Berger,Severine Morisset-Lopez, Francois Lefoulon,Carlo Pifferi,Vincent Aucagne

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY(2023)

引用 0|浏览16
关键词
Chemical biology,Drug synergy,Native chemical ligation,Peptide,Protein-drug conjugate,Synthetic protein
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