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Discovery of Pyrazolopyrazines As Selective, Potent, and Mutant-Active MET Inhibitors with Intracranial Efficacy

Quinn A. Bumpers,Robert W. Pipal, Anna M. Benz-Weeden,James T. Brewster II, Adam Cook, Amy L. Crooks,Cole Cruz,Natalie C. Dwulet,John J. Gaudino, Daniel Golec, Jacqueline A. Harrison,Dylan P. Hartley, Sherif H. Hassanien,Erik J. Hicken, Dean Kahn,Ellen R. Laird,Christine Lemieux, Nicholas Lewandowski, Joseph Mccown,Matthew G. Mcdonald, Oren Mcnulty,Tung-Chung Mou, Phong Nguyen, Lauren Oko, Lisa Pieti Opie,Jennifer Otten,Spencer C. Peck,Viktor C. Polites, Samuel D. Randall, Rachel Z. Rosen,Pavel Savechenkov, Helen Simpson,Anurag Singh, Drew Sparks, Kyle Wickersham,Lance Wollenberg,Christina E. Wong,Jim Wong, Wen- Wu,Mohamed S. A. Elsayed,Ronald J. Hinklin,Tony P. Tang

Journal of Medicinal Chemistry(2024)

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