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Application of a Macrocyclization Strategy in Kinase Inhibitor Development

Kun Xing, Shujun Li, Jinghuan Li,Dan Liu,Min Huang, Linxiang Zhao

Acta Materia Medica(2025)

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关键词
kinase inhibitor,macrocyclization strategy,drug design,binding affinity,kinase selectivity,drug-like properties
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