Darryl S. Pickering - Faculty of Pharmaceutical Sciences, University of Copenhagen

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论文共 160 篇作者统计合作学者相似作者

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Exploring Thienothiadiazine Dioxides As Isosteric Analogues of Benzo- and Pyridothiadiazine Dioxides in the Search of New AMPA and Kainate Receptor Positive Allosteric Modulators

Pierre Francotte,Yasmin Bay,Eric Goffin,Thomas Colson, Cindy Lesenfants,Jerzy Dorosz,Saara Laulumaa,Pierre Fraikin,Pascal de Tullio, Caroline Beaufour,Iuliana Botez,Darryl S. Pickering,Karla Frydenvang,Laurence Danober,Anders Skov Kristensen,Jette Sandholm Kastrup,Bernard Pirotte

EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY（2024）

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Small Molecule Positive Allosteric Modulation of Homomeric Kainate Receptors GluK1-3: Development of Screening Assays and Insight into GluK3 Structure

Yasmin Bay,Raminta Venskutonyte,Stine M. Frantsen,Thor S. Thorsen,Maria Musgaard,Karla Frydenvang,Pierre Francotte,Bernard Pirotte,Philip C. Biggin,Anders S. Kristensen,Thomas Boesen,Darryl S. Pickering,Michael Gajhede,Jette S. Kastrup

FEBS JOURNAL（2024）

引用1浏览0WOS引用

Domoic Acid As a Lead for the Discovery of the First Selective Ligand for Kainate Receptor Subtype 5 (Gluk5)

Silke Buschbom-Helmke, Pengfei Wang,Anna Alcaide,Federico Miguez-Cabello,Mario Carta, Julio S. Viotti,Birgitte Nielsen,Christophe Mulle,Derek Bowie,Flemming Steen Jorgensen,Darryl S. Pickering,Lennart Bunch

Journal of Medicinal Chemistryno. 16 (2024): 14524-14542

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Active-like Structure of the Ligand-Binding Domain of GluK2 with L-glutamate and the Positive Allosteric Modulator BPAM344

Yasmin Bay, Mie Egeberg Jeppesen,Karla Frydenvang,Pierre Francotte,Bernard Pirotte,Darryl S. Pickering,Anders Skov Kristensen,Jette Sandholm Kastrup

FEBS Letters (2024)

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Tritium and Deuterium Labelling of a Kainate Receptor Antagonist and Evaluation As a Radioligand

Paulina Chalupnik,Ales Marek, Marie Emilie Leiticia Hovah,Darryl S. Pickering,Piero Temperini, Stephanie Donbosco,Ewa Szymanska,Tommy N. Johansen

Journal of Labelled Compounds and Radiopharmaceuticalsno. 4 (2024): 120-130

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Crystal Structure of the GluK1 Ligand-Binding Domain with Kainate and the Full-Spanning Positive Allosteric Modulator BPAM538

Yasmin Bay, Federico Javier Miguez Cabello, Chloe C. Koens,Stine M. Frantsen,Darryl S. Pickering,Karla Frydenvang,Pierre Francotte,Bernard Pirotte,Anders S. Kristensen,Derek Bowie,Jette Sandholm Kastrup

JOURNAL OF STRUCTURAL BIOLOGY（2024）

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Structure-Activity Relationship and Solubility Studies of N1-Substituted Quinoxaline-2,3-diones As Kainate Receptor Antagonists

Paulina Chalupnik,Alina Vialko,Darryl S. Pickering,Birgitte Nielsen,Yasmin Bay,Anders Skov Kristensen,Markus Hinkkanen,Katarzyna Szczepanska,Tadeusz Karcz,Gniewomir Latacz,Tommy N. Johansen,Ewa Szymanska

CHEMMEDCHEMno. 18 (2023)

引用2浏览0WOS引用

Discovery of the First Highly Selective Antagonist of the GluK3 Kainate Receptor Subtype

Paulina Chalupnik,Alina Vialko,Darryl S. Pickering,Markus Hinkkanen, Stephanie Donbosco,Thor C. Moller,Anders A. Jensen,Birgitte Nielsen,Yasmin Bay,Anders S. Kristensen,Tommy N. Johansen,Kamil Latka,Marek Bajda,Ewa Szymanska

International Journal of Molecular Sciences（2022）

引用6浏览0WOS引用

(S)-2-mercaptohistidine: A First Selective Orthosteric GluK3 Antagonist

Christian B. M. Poulie,Younes Larsen,Cindie Leteneur,Gael Barthet,Walden E. Bjorn-Yoshimoto,Fanny Malhaire,Birgitte Nielsen, Jean-Phillippe Pin,Christophe Mulle,Darryl S. Pickering,Lennart Bunch

ACS chemical neuroscience（2022）

引用2浏览0WOS引用

Structural Basis for Positive Allosteric Modulation of AMPA and Kainate Receptors

Karla Frydenvang,Darryl S. Pickering,Jette Sandholm Kastrup

The Journal of Physiology（2021）

引用12浏览0WOS引用

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